Compile Data Set for Download or QSAR
maximum 50k data
Found 5 of ec50 data for polymerid = 50004796
TargetTransmembrane protease serine 2(Homo sapiens (Human))
Shionogi

LigandPNGBDBM513874(bioRxiv20220126.477782, S-217622 | bioRxiv20220126...)
Affinity DataEC50:  370nMAssay Description:Antiviral activity against SARS-CoV-2, SARS-CoV, MERS-CoV and HCoV-229E was assessed by monitoring cell viability; that against HCoV-OC43 was assesse...More data for this Ligand-Target Pair
In DepthDetails
TargetTransmembrane protease serine 2(Homo sapiens (Human))
Shionogi

LigandPNGBDBM50424712(CAMOSTAT | Camostat Mesilate | Foipan)
Affinity DataEC50:  1.00E+3nMAssay Description:Inhibition of human TMPRSS2-mediated SARS-CoV-2 entry into human Caco-2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransmembrane protease serine 2(Homo sapiens (Human))
Shionogi

LigandPNGBDBM50031706(4-Guanidino-benzoic acid 4-dimethylcarbamoylmethox...)
Affinity DataEC50:  1.00E+4nMAssay Description:This is a review article.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransmembrane protease serine 2(Homo sapiens (Human))
Shionogi

LigandPNGBDBM513873(bioRxiv20220126.477782, Screening Hit 2)
Affinity DataEC50:  1.25E+4nMAssay Description:Antiviral activity against SARS-CoV-2, SARS-CoV, MERS-CoV and HCoV-229E was assessed by monitoring cell viability; that against HCoV-OC43 was assesse...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetTransmembrane protease serine 2(Homo sapiens (Human))
Shionogi

LigandPNGBDBM533518(jm2c00120, Compound 17)
Affinity DataEC50:  8.40E+4nMAssay Description:Ec50 of SARS-CoV-infected VeroE6 cells.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed